检索结果 - David C. Dalgarno
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Activity of dual SRC-ABL inhibitors highlights the role of BCR/ABL kinase dynamics in drug resistance 由 Mohammad Azam, Valentina Nardi, William C. Shakespeare, Chester A. Metcalf, Regine S. Bohacek, Yihan Wang, Raji Sundaramoorthi, Piotr Sliz, Darren R. Veach, William G. Bornmann, Bayard Clarkson, David C. Dalgarno, Tomi K. Sawyer, George Q. Daley
出版 2006Artigo -
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Crizotinib‐Resistant Mutants of EML4‐ALK Identified Through an Accelerated Mutagenesis Screen 由 Sen Zhang, Frank Wang, Jeffrey Keats, Xiaotian Zhu, Yaoyu Ning, Scott Wardwell, Lauren Moran, Qurish K. Mohemmad, Rana Anjum, Yihan Wang, Narayana I. Narasimhan, David C. Dalgarno, William C. Shakespeare, Juan J. Miret, Tim Clackson, Victor M. Rivera
出版 2011Carta -
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Inhibition of wild-type and mutant Bcr-Abl by AP23464, a potent ATP-based oncogenic protein kinase inhibitor: implications for CML 由 Thomas O’Hare, Roy M. Pollock, Eric P. Stoffregen, Jeffrey Keats, Omar Mohammed Abdullah, Erika M. Mosesón, Victor M. Rivera, Hao Tang, Chester A. Metcalf, Regine S. Bohacek, Yihan Wang, Raji Sundaramoorthi, William C. Shakespeare, David C. Dalgarno, Tim Clackson, Tomi K. Sawyer, Michael W. Deininger, Brian J. Druker
出版 2004Artigo -
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Structural Basis of Src Tyrosine Kinase Inhibition with a New Class of Potent and Selective Trisubstituted Purine‐based Compounds 由 David C. Dalgarno, Thilo Stehle, Surinder S. Narula, P. Schelling, Marie Rose van Schravendijk, Susan Adams, Lawrence Andrade, Jeff Keats, Mary K. Ram, Lei Jin, Trudy H. Grossman, Ian A. MacNeil, Chester A. Metcalf, William C. Shakespeare, Yihan Wang, Terry Keenan, Raji Sundaramoorthi, Regine S. Bohacek, Manfred Weigele, Tomi K. Sawyer
出版 2005Artigo -
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Antiangiogenic and Antitumor Effects of Src Inhibition in Ovarian Carcinoma 由 Liz Y. Han, Charles N. Landen, José G. Treviño, Jyotsnabaran Halder, Yvonne G. Lin, Aparna A. Kamat, Tae‐Jin Kim, William M. Merritt, Robert L. Coleman, David M. Gershenson, William C. Shakespeare, Yihan Wang, Raji Sundaramoorth, Chester A. Metcalf, David C. Dalgarno, Tomi K. Sawyer, Gary E. Gallick, Anil K. Sood
出版 2006Artigo -
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Mobocertinib (TAK-788): A Targeted Inhibitor of<i>EGFR</i>Exon 20 Insertion Mutants in Non–Small Cell Lung Cancer 由 Francois Gonzalvez, Sylvie Vincent, Theresa E. Baker, Alexandra E. Gould, Shuai Li, Scott Wardwell, Sara Nadworny, Yaoyu Ning, Sen Zhang, Wei‐Sheng Huang, Yongbo Hu, Feng Li, Matthew T. Greenfield, Stephan G. Zech, Biplab Das, Narayana I. Narasimhan, Tim Clackson, David C. Dalgarno, William C. Shakespeare, Michael Fitzgerald, Johara Chouitar, Robert Griffin, Shengwu Liu, Kwok‐Kin Wong, Xiaotian Zhu, Victor M. Rivera
出版 2021Artigo -
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AP24534, a Pan-BCR-ABL Inhibitor for Chronic Myeloid Leukemia, Potently Inhibits the T315I Mutant and Overcomes Mutation-Based Resistance 由 Thomas O’Hare, William C. Shakespeare, Xiaotian Zhu, Christopher A. Eide, Victor M. Rivera, Frank Wang, Lauren T. Adrian, Tianjun Zhou, Wei-Sheng Huang, Qihong Xu, Chester A. Metcalf, Jeffrey W. Tyner, Marc Loriaux, Amie S. Corbin, Scott Wardwell, Yaoyu Ning, Jeffrey Keats, Yihan Wang, Raji Sundaramoorthi, Mathew Thomas, Dong Zhou, J. T. Snodgrass, Lois Commodore, Tomi K. Sawyer, David C. Dalgarno, Michael W. Deininger, Brian J. Druker, Tim Clackson
出版 2009Artigo -
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Structure-based design of an osteoclast-selective, nonpeptide Src homology 2 inhibitor with <i>in vivo</i> antiresorptive activity 由 William C. Shakespeare, Michael G. Yang, Regine S. Bohacek, Franklin Cerasoli, Karin J. Stebbins, Raji Sundaramoorthi, Mihai Azimioara, Chi B. Vu, Selvi Pradeepan, Chester A. Metcalf, Chad A. Haraldson, Taylor Merry, David C. Dalgarno, Surinder S. Narula, Marcos Hatada, Xiaode Lu, Marie Rose van Schravendijk, Susan Adams, Shelia M. Violette, Jeremy A. Smith, Wei Guan, Catherine Bartlett, Jay Herson, John D. Iuliucci, Manfred Weigele, Tomi K. Sawyer
出版 2000Artigo -
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The Potent ALK Inhibitor Brigatinib (AP26113) Overcomes Mechanisms of Resistance to First- and Second-Generation ALK Inhibitors in Preclinical Models 由 Sen Zhang, Rana Anjum, Rachel M. Squillace, Sara Nadworny, Tianjun Zhou, Jeff Keats, Yaoyu Ning, Scott Wardwell, David F. Miller, Youngchul Song, Lindsey Eichinger, Lauren Moran, Wei‐Sheng Huang, Shuangying Liu, Dong Zou, Yihan Wang, Qurish K. Mohemmad, Hyun Gyung Jang, Emily Ye, Narayana I. Narasimhan, Frank Wang, Juan J. Miret, Xiaotian Zhu, Tim Clackson, David C. Dalgarno, William C. Shakespeare, Victor M. Rivera
出版 2016Artigo
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Biology
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Proto-oncogene tyrosine-protein kinase Src
Tyrosine kinase
ABL
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ALK inhibitor
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Crizotinib
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