نتائج البحث - David C. Dalgarno
- يعرض 1 - 12 نتائج من 12
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Activity of dual SRC-ABL inhibitors highlights the role of BCR/ABL kinase dynamics in drug resistance حسب Mohammad Azam, Valentina Nardi, William C. Shakespeare, Chester A. Metcalf, Regine S. Bohacek, Yihan Wang, Raji Sundaramoorthi, Piotr Sliz, Darren R. Veach, William G. Bornmann, Bayard Clarkson, David C. Dalgarno, Tomi K. Sawyer, George Q. Daley
منشور في 2006Artigo -
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Crizotinib‐Resistant Mutants of EML4‐ALK Identified Through an Accelerated Mutagenesis Screen حسب Sen Zhang, Frank Wang, Jeffrey Keats, Xiaotian Zhu, Yaoyu Ning, Scott Wardwell, Lauren Moran, Qurish K. Mohemmad, Rana Anjum, Yihan Wang, Narayana I. Narasimhan, David C. Dalgarno, William C. Shakespeare, Juan J. Miret, Tim Clackson, Victor M. Rivera
منشور في 2011Carta -
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Inhibition of wild-type and mutant Bcr-Abl by AP23464, a potent ATP-based oncogenic protein kinase inhibitor: implications for CML حسب Thomas O’Hare, Roy M. Pollock, Eric P. Stoffregen, Jeffrey Keats, Omar Mohammed Abdullah, Erika M. Mosesón, Victor M. Rivera, Hao Tang, Chester A. Metcalf, Regine S. Bohacek, Yihan Wang, Raji Sundaramoorthi, William C. Shakespeare, David C. Dalgarno, Tim Clackson, Tomi K. Sawyer, Michael W. Deininger, Brian J. Druker
منشور في 2004Artigo -
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Structural Basis of Src Tyrosine Kinase Inhibition with a New Class of Potent and Selective Trisubstituted Purine‐based Compounds حسب David C. Dalgarno, Thilo Stehle, Surinder S. Narula, P. Schelling, Marie Rose van Schravendijk, Susan Adams, Lawrence Andrade, Jeff Keats, Mary K. Ram, Lei Jin, Trudy H. Grossman, Ian A. MacNeil, Chester A. Metcalf, William C. Shakespeare, Yihan Wang, Terry Keenan, Raji Sundaramoorthi, Regine S. Bohacek, Manfred Weigele, Tomi K. Sawyer
منشور في 2005Artigo -
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Antiangiogenic and Antitumor Effects of Src Inhibition in Ovarian Carcinoma حسب Liz Y. Han, Charles N. Landen, José G. Treviño, Jyotsnabaran Halder, Yvonne G. Lin, Aparna A. Kamat, Tae‐Jin Kim, William M. Merritt, Robert L. Coleman, David M. Gershenson, William C. Shakespeare, Yihan Wang, Raji Sundaramoorth, Chester A. Metcalf, David C. Dalgarno, Tomi K. Sawyer, Gary E. Gallick, Anil K. Sood
منشور في 2006Artigo -
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Mobocertinib (TAK-788): A Targeted Inhibitor of<i>EGFR</i>Exon 20 Insertion Mutants in Non–Small Cell Lung Cancer حسب Francois Gonzalvez, Sylvie Vincent, Theresa E. Baker, Alexandra E. Gould, Shuai Li, Scott Wardwell, Sara Nadworny, Yaoyu Ning, Sen Zhang, Wei‐Sheng Huang, Yongbo Hu, Feng Li, Matthew T. Greenfield, Stephan G. Zech, Biplab Das, Narayana I. Narasimhan, Tim Clackson, David C. Dalgarno, William C. Shakespeare, Michael Fitzgerald, Johara Chouitar, Robert Griffin, Shengwu Liu, Kwok‐Kin Wong, Xiaotian Zhu, Victor M. Rivera
منشور في 2021Artigo -
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AP24534, a Pan-BCR-ABL Inhibitor for Chronic Myeloid Leukemia, Potently Inhibits the T315I Mutant and Overcomes Mutation-Based Resistance حسب Thomas O’Hare, William C. Shakespeare, Xiaotian Zhu, Christopher A. Eide, Victor M. Rivera, Frank Wang, Lauren T. Adrian, Tianjun Zhou, Wei-Sheng Huang, Qihong Xu, Chester A. Metcalf, Jeffrey W. Tyner, Marc Loriaux, Amie S. Corbin, Scott Wardwell, Yaoyu Ning, Jeffrey Keats, Yihan Wang, Raji Sundaramoorthi, Mathew Thomas, Dong Zhou, J. T. Snodgrass, Lois Commodore, Tomi K. Sawyer, David C. Dalgarno, Michael W. Deininger, Brian J. Druker, Tim Clackson
منشور في 2009Artigo -
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Structure-based design of an osteoclast-selective, nonpeptide Src homology 2 inhibitor with <i>in vivo</i> antiresorptive activity حسب William C. Shakespeare, Michael G. Yang, Regine S. Bohacek, Franklin Cerasoli, Karin J. Stebbins, Raji Sundaramoorthi, Mihai Azimioara, Chi B. Vu, Selvi Pradeepan, Chester A. Metcalf, Chad A. Haraldson, Taylor Merry, David C. Dalgarno, Surinder S. Narula, Marcos Hatada, Xiaode Lu, Marie Rose van Schravendijk, Susan Adams, Shelia M. Violette, Jeremy A. Smith, Wei Guan, Catherine Bartlett, Jay Herson, John D. Iuliucci, Manfred Weigele, Tomi K. Sawyer
منشور في 2000Artigo -
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The Potent ALK Inhibitor Brigatinib (AP26113) Overcomes Mechanisms of Resistance to First- and Second-Generation ALK Inhibitors in Preclinical Models حسب Sen Zhang, Rana Anjum, Rachel M. Squillace, Sara Nadworny, Tianjun Zhou, Jeff Keats, Yaoyu Ning, Scott Wardwell, David F. Miller, Youngchul Song, Lindsey Eichinger, Lauren Moran, Wei‐Sheng Huang, Shuangying Liu, Dong Zou, Yihan Wang, Qurish K. Mohemmad, Hyun Gyung Jang, Emily Ye, Narayana I. Narasimhan, Frank Wang, Juan J. Miret, Xiaotian Zhu, Tim Clackson, David C. Dalgarno, William C. Shakespeare, Victor M. Rivera
منشور في 2016Artigo
أدوات البحث:
موضوعات ذات صلة
Biology
Cancer research
Gene
Biochemistry
Chemistry
Genetics
Mutation
Signal transduction
Kinase
Medicine
Mutant
Proto-oncogene tyrosine-protein kinase Src
Tyrosine kinase
ABL
Cancer
Lung cancer
Myeloid leukemia
Pharmacology
ALK inhibitor
Alectinib
Anaplastic lymphoma kinase
Astronomy
Crizotinib
Crystallography
Imatinib
Imatinib mesylate
In vivo
Internal medicine
Malignant pleural effusion
Mutagenesis