検索結果 - Daniel Robbins
- 検索結果 1 - 9 結果 / 9
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Nx-5948, a Selective Degrader of BTK with Activity in Preclinical Models of Hematologic and Brain Malignancies 著者: Daniel Robbins, Mark Noviski, Ryan B. Rountree, May Tan, Nivetha Brathaban, Timothy Ingallinera, Dane E. Karr, Aileen Kelly, Zef Konst, Jun Ma, Austin Tenn-McClellan, Jenny McKinnell, Luz Perez, Cristiana Guiducci, Gwenn M. Hansen, Arthur Sands
出版事項 2021Artigo -
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Nx-2127, a Degrader of BTK and IMiD Neosubstrates, for the Treatment of B-Cell Malignancies 著者: Daniel Robbins, Aileen Kelly, May Tan, Joel McIntosh, Jeffrey Wu, Zef Konst, Daisuke Kato, Ge Peng, Jeff Mihalic, Dahlia R. Weiss, Luz Perez, Jennifer Tung, Anna Kolobova, Sasha Borodovsky, Ryan B. Rountree, Austin Tenn-McClellan, Mark Noviski, Jordan Ye, Stephen E. Basham, Timothy Ingallinera, Jenny McKinnell, Dane E. Karr, Janine Powers, Cristiana Guiducci, Arthur Sands
出版事項 2020Artigo -
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Discovery and Preclinical Pharmacology of NX-2127, an Orally Bioavailable Degrader of Bruton’s Tyrosine Kinase with Immunomodulatory Activity for the Treatment of Patients with B C... 著者: Daniel Robbins, Mark Noviski, Ying Siow Tan, Zef A. Könst, Aileen Kelly, P Auger, Nivetha Brathaban, Robert Cass, Ming Liang Chan, Ganesh Cherala, Matthew C. Clifton, Stefan Gajewski, Timothy G. Ingallinera, Dane E. Karr, Daisuke Kato, Jun Ma, Jenny McKinnell, Joel McIntosh, Jeff Mihalic, Brent Murphy, Panga Jaipal Reddy, Ge Peng, Janine Powers, Luz Perez, Ryan B. Rountree, Austin Tenn-McClellan, Arthur Sands, Dahlia R. Weiss, Jeffrey Wu, Jordan Ye, Cristiana Guiducci, Gwenn M. Hansen, Frederick Cohen
出版事項 2024Artigo -
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Structure Based Design of Non-Natural Peptidic Macrocyclic Mcl-1 Inhibitors 著者: Jeffrey W. Johannes, Stephanie M. Bates, Carl Beigie, Matthew A. Belmonte, John Breen, Shenggen Cao, Paolo A. Centrella, Matthew Clark, John W. Cuozzo, Christoph E. Dumelin, Andrew D. Ferguson, Sevan Habeshian, David Hargreaves, Camil Joubran, Steven L. Kazmirski, Anthony D. Keefe, Michelle L. Lamb, Haiye Lan, Yunxia Li, Hao Ma, Scott N. Mlynarski, Martin J. Packer, Philip B. Rawlins, Daniel Robbins, Haidong Shen, Eric A. Sigel, Holly H. Soutter, Nancy Su, Dawn M. Troast, Haiyun Wang, Kate F. Wickson, Chengyan Wu, Ying Zhang, Qiuying Zhao, Xiaolan Zheng, Alexander W. Hird
出版事項 2016Artigo -
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Discovery of Mcl-1-specific inhibitor AZD5991 and preclinical activity in multiple myeloma and acute myeloid leukemia 著者: Adriana E. Tron, Matthew A. Belmonte, Ammar Adam, Brian Aquila, Lawrence Boise, Elisabetta Chiarparin, Justin Cidado, Kevin J. Embrey, Eric T. Gangl, Francis D. Gibbons, Gareth P. Gregory, David Hargreaves, J. Adam Hendricks, Jeffrey W. Johannes, Ricky W. Johnstone, Steven L. Kazmirski, Jason G. Kettle, Michelle L. Lamb, Shannon M. Matulis, Ajay K. Nooka, Martin J. Packer, Bo Peng, Philip B. Rawlins, Daniel Robbins, Alwin G. Schuller, Nancy Su, Wenzhan Yang, Qing Ye, Xiaolan Zheng, J. Paul Secrist, Edwin Clark, David M. Wilson, Stephen E. Fawell, Alexander W. Hird
出版事項 2018Artigo
関連主題
Medicine
Biology
Chemistry
Biochemistry
Cancer research
Chronic lymphocytic leukemia
Immunology
Internal medicine
Leukemia
Bruton's tyrosine kinase
Computer science
Ibrutinib
Physical medicine and rehabilitation
Physical therapy
Physics
Psychology
Signal transduction
Tyrosine kinase
Agonist
Agonist-antagonist
Antagonist
Combinatorial chemistry
Gene
Pharmacology
Receptor
Resistance training
Ubiquitin
Ubiquitin ligase
Acceleration
Acoustics