Resultats de la cerca - Cosimo G. Fortuna
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1
Structural basis for selective inhibition of Cyclooxygenase-1 (COX-1) by diarylisoxazoles mofezolac and 3-(5-chlorofuran-2-yl)-5-methyl-4-phenylisoxazole (P6) per Gino Cingolani, Andrea Panella, Maria Grazia Perrone, Paola Vitale, Giuseppe Di Mauro, Cosimo G. Fortuna, Roger S. Armen, Savina Ferorelli, William L. Smith, Antonio Scilimati
Publicat 2017Artigo -
2
A further pocket or conformational plasticity by mapping COX-1 catalytic site through modified-mofezolac structure-inhibitory activity relationships and their antiplatelet behavior per Roberta Solidoro, Morena Miciaccia, Carmela Bonaccorso, Cosimo G. Fortuna, Domenico Armenise, Antonella Centonze, Savina Ferorelli, Paola Vitale, Pryscila Rodrigues, Renilda Guimarães, Alana de Oliveira, Mariana da Paz, Luciana P. Rangel, P.C Sathler, Angela Altomare, Maria Grazia Perrone, Antonio Scilimati
Publicat 2024Artigo -
3
Harmaline to Human Mitochondrial Caseinolytic Serine Protease Activation for Pediatric Diffuse Intrinsic Pontine Glioma Treatment per Morena Miciaccia, Francesca Rizzo, Antonella Centonze, Gianfranco Cavallaro, Marialessandra Contino, Domenico Armenise, Olga Maria Baldelli, Roberta Solidoro, Savina Ferorelli, Pasquale Scarcia, Gennaro Agrimi, Veronica Zingales, Elisa Cimetta, Simone Ronsisvalle, Federica Sipala, Paola Loguercio Polosa, Cosimo G. Fortuna, Maria Grazia Perrone, Antonio Scilimati
Publicat 2024Artigo
Eines de cerca:
Matèries relacionades
Biochemistry
Chemistry
Active site
Cyclooxygenase
Enzyme
Enzyme inhibitor
In vitro
Stereochemistry
Structure–activity relationship
Alkyl
Apoptosis
Binding site
Biology
Cancer research
Catalysis
Cell
Cell biology
Context (archaeology)
Crystal structure
Crystallography
Enzyme kinetics
Halogen
Harmaline
IC50
Isopropyl
Isoxazole
Medicinal chemistry
Medicine
Mitochondrion
Moiety