Search Results - Christophe Dardonville
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New Bis(2-aminoimidazoline) and Bisguanidine DNA Minor Groove Binders with Potent in Vivo Antitrypanosomal and Antiplasmodial Activity by Fernando Rodrı́guez, Isabel Rozas, Marcel Kaiser, Reto Brun, Binh Nguyen, W. David Wilson, Rory Nelson García, Christophe Dardonville
Published 2008Artigo -
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Nanostructured Lipid Carrier for Intracellular Delivery of a Bis(pyridine-2-carboxamidine) DNA Minor Groove Binder Active against <i>Leishmania</i> by J. Jonathan Nué-Martínez, Marta Leo-Barriga, Fernando Herranz, Zisis Koutsogiannis, Paul W. Denny, Godwin U. Ebiloma, Christophe Dardonville, Ana González-Paredes
Published 2025Artigo -
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Synthesis and Structure–Activity Analysis of New Phosphonium Salts with Potent Activity against African Trypanosomes by Andrea Taladriz‐Sender, Alan R. Healy, Eddysson J. Flores Pérez, Vanessa Herrero, Carlos Ríos-Martínez, Abdulsalam A. M. Alkhaldi, Anthonius A. Eze, Marcel Kaiser, Harry P. de Koning, Antonio Chana, Christophe Dardonville
Published 2012Artigo -
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Positively selected modifications in the pore of TbAQP2 allow pentamidine to enter Trypanosoma brucei by Ali Al-Ghamdi, Jane C. Munday, Gustavo D. Campagnaro, Dominik Gurvič, Fredrik Svensson, Chinyere E. Okpara, Arvind Kumar, Juan F. Quintana, Maria Esther Martin Abril, Patrik Milić, Laura N. Watson, Daniel Paape, Luca Settimo, Anna Dimitriou, Joanna Wielińska, Graeme Smart, Laura Anderson, Christopher M. Woodley, Siu Pui Ying Kelly, Hasan M. S. Ibrahim, Fabian Hulpia, Mohammed I. Al‐Salabi, Anthonius A. Eze, Teresa Sprenger, Ibrahim A. Teka, Simon Gudin, Simone Weyand, Mark C. Field, Christophe Dardonville, Richard R. Tidwell, Mark Carrington, Paul M. O’Neill, David W. Boykin, Ulrich Zachariae, Harry P. de Koning
Published 2020Artigo
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Biochemistry
Biology
Chemistry
Gene
Trypanosoma brucei
DNA
In vitro
Mitochondrion
Organic chemistry
Pharmacology
Stereochemistry
Biophysics
Cell biology
Enzyme
Genetics
Mechanism of action
Medicine
Pentamidine
Pneumonia
Structure–activity relationship
Transporter
Trypanosoma brucei rhodesiense
ATPase
Alternative oxidase
Antiparasitic
Archaeology
Benzophenone
Combinatorial chemistry
Groove (engineering)
Guanidine