Výsledky vyhledávání - Chris Phillips
- Zobrazuji výsledky 1 - 9 z 9
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Discovery of a novel allosteric inhibitor-binding site in ERK5: comparison with the canonical kinase hinge ATP-binding site Autor Hongming Chen, Julie A. Tucker, Xiaotao Wang, Paul R. Gavine, Chris Phillips, Martin Augustin, Patrick Schreiner, Stefan Steinbacher, Marian Preston, D. Ogg
Vydáno 2016Artigo -
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Structural basis of Lewis <sup>b</sup> antigen binding by the <i>Helicobacter pylori</i> adhesin BabA Autor Naim Hage, Tina Howard, Chris Phillips, C. Brassington, R. Overman, J.E. Debreczeni, Paul Gellert, Snow Stolnik, G. Sebastiaan Winkler, Franco H. Falcone
Vydáno 2015Artigo -
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Lersivirine, a Nonnucleoside Reverse Transcriptase Inhibitor with Activity against Drug-Resistant Human Immunodeficiency Virus Type 1 Autor Romuald Corbau, Julie Mori, Chris Phillips, Lesley Fishburn, Alex Martín, Charles E. Mowbray, Wendy Panton, Caroline Smith‐Burchnell, Adele Thornberry, H. Ringrose, Thorsten Knöchel, Steve Irving, Mike Westby, Anthony Wood, Manos Perros
Vydáno 2010Artigo -
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Structural and dynamic insights into the energetics of activation loop rearrangement in FGFR1 kinase Autor Tobias Klein, Navratna Vajpai, Jonathan J. Phillips, Gareth M. Davies, Geoffrey A. Holdgate, Chris Phillips, Julie A. Tucker, Richard A. Norman, Andrew D. Scott, Daniel R. Higazi, David C. Lowe, Gary S. Thompson, Alexander L. Breeze
Vydáno 2015Artigo -
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Cryo-EM structure determination of small therapeutic protein targets at 3 Å-resolution using a rigid imaging scaffold Autor Roger Castells‐Graells, Kyle Meador, Mark A. Arbing, M.R. Sawaya, Morgan Gee, Duilio Cascio, Emma S. Gleave, J.E. Debreczeni, J. Breed, Karoline Leopold, Ankoor Patel, Dushyant Jahagirdar, Bronwyn Lyons, Sriram Subramaniam, Chris Phillips, Todd O. Yeates
Vydáno 2023Artigo -
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Landscape of activating cancer mutations in FGFR kinases and their differential responses to inhibitors in clinical use Autor Harshnira Hitesh Patani, Tom D. Bunney, Nethaji Thiyagarajan, Richard A. Norman, D. Ogg, J. Breed, Paul Ashford, Andrew Potterton, Mina Edwards, Sarah V. Williams, Gary S. Thomson, Camilla Pang, Margaret A. Knowles, Alexander L. Breeze, Christine Orengo, Chris Phillips, Matilda Katan
Vydáno 2016Artigo -
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Recurrent MLK4 Loss-of-Function Mutations Suppress JNK Signaling to Promote Colon Tumorigenesis Autor Anna A. Marusiak, Natalie L. Stephenson, Hayeon Baik, Eleanor W. Trotter, Yaoyong Li, Karen Blyth, Susan Mason, Phil Chapman, Lorena A. Puto, Jon Read, C. Brassington, Hannah Pollard, Chris Phillips, Isabelle Green, R. Overman, Matthew Collier, Ewelina Testoni, Crispin Miller, Tony Hunter, Owen J. Sansom, John Brognard
Vydáno 2015Artigo
Vyhledávací nástroje:
Související témata
Biology
Gene
Biochemistry
Chemistry
Drug discovery
Genetics
Medicine
Mutant
Computational biology
Kinase
Mutation
Receptor
Binding site
Bioinformatics
Biophysics
Cancer research
Computer science
Drug
Fibroblast growth factor
Human immunodeficiency virus (HIV)
Pharmacology
Protein kinase domain
RNA
Reverse transcriptase
Signal transduction
Virology
Allosteric enzyme
Allosteric regulation
Antigen
Antiretroviral therapy