Результаты поиска - Azuaje, Jhonny
- Отображение 1 - 9 результаты of 9
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Computer-aided design of multi-target ligands at A(1)R, A(2A)R and PDE10A, key proteins in neurodegenerative diseases по Kalash, Leen, Val, Cristina, Azuaje, Jhonny, Loza, María I., Svensson, Fredrik, Zoufir, Azedine, Mervin, Lewis, Ladds, Graham, Brea, José, Glen, Robert, Sotelo, Eddy, Bender, Andreas
Опубликовано 2017Текст -
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Discovery of 3,4-Dihydropyrimidin-2(1H)-ones As a Novel Class of Potent and Selective A(2B) Adenosine Receptor Antagonists по Crespo, Abel, El Maatougui, Abdelaziz, Biagini, Pierfrancesco, Azuaje, Jhonny, Coelho, Alberto, Brea, José, Loza, María Isabel, Cadavid, María Isabel, García-Mera, Xerardo, Gutiérrez-de-Terán, Hugo, Sotelo, Eddy
Опубликовано 2013Текст -
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Potent and Subtype-Selective Dopamine D(2) Receptor Biased Partial Agonists Discovered via an Ugi-Based Approach по Mallo-Abreu, Ana, Reyes-Resina, Irene, Azuaje, Jhonny, Franco, Rafael, García-Rey, Aitor, Majellaro, Maria, Miranda-Pastoriza, Darío, García-Mera, Xerardo, Jespers, Willem, Gutiérrez-de-Terán, Hugo, Navarro, Gemma, Sotelo, Eddy
Опубликовано 2021Текст -
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Development of Fluorescent Probes that Target Serotonin 5-HT(2B) Receptors по Azuaje, Jhonny, López, Paula, Iglesias, Alba, de la Fuente, Rocío A., Pérez-Rubio, José M., García, Diego, Stępniewski, Tomasz Maciej, García-Mera, Xerardo, Brea, José M., Selent, Jana, Pérez, Dolores, Castro, Marián, Loza, María I., Sotelo, Eddy
Опубликовано 2017Текст -
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X‐Ray Crystallography and Free Energy Calculations Reveal the Binding Mechanism of A(2A) Adenosine Receptor Antagonists по Jespers, Willem, Verdon, Grégory, Azuaje, Jhonny, Majellaro, Maria, Keränen, Henrik, García‐Mera, Xerardo, Congreve, Miles, Deflorian, Francesca, de Graaf, Chris, Zhukov, Andrei, Doré, Andrew S., Mason, Jonathan S., Åqvist, Johan, Cooke, Robert M., Sotelo, Eddy, Gutiérrez‐de‐Terán, Hugo
Опубликовано 2020Текст -
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Exploring Non-orthosteric Interactions with a Series of Potent and Selective A(3) Antagonists по Miranda-Pastoriza, Darío, Bernárdez, Rodrigo, Azuaje, Jhonny, Prieto-Díaz, Rubén, Majellaro, Maria, Tamhankar, Ashish V., Koenekoop, Lucien, González, Alejandro, Gioé-Gallo, Claudia, Mallo-Abreu, Ana, Brea, José, Loza, M. Isabel, García-Rey, Aitor, García-Mera, Xerardo, Gutiérrez-de-Terán, Hugo, Sotelo, Eddy
Опубликовано 2022Текст -
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Optimization of 2-Amino-4,6-diarylpyrimidine-5-carbonitriles as Potent and Selective A(1) Antagonists по Val, Cristina, Rodríguez-García, Carlos, Prieto-Díaz, Rubén, Crespo, Abel, Azuaje, Jhonny, Carbajales, Carlos, Majellaro, Maria, Díaz-Holguín, Alejandro, Brea, José M., Loza, Maria Isabel, Gioé-Gallo, Claudia, Contino, Marialessandra, Stefanachi, Angela, García-Mera, Xerardo, Estévez, Juan C., Gutiérrez-de-Terán, Hugo, Sotelo, Eddy
Опубликовано 2022Текст -
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A(2B) adenosine receptor antagonists rescue lymphocyte activity in adenosine-producing patient-derived cancer models по Tay, Apple Hui Min, Prieto-Díaz, Rubén, Neo, Shiyong, Tong, Le, Chen, Xinsong, Carannante, Valentina, Önfelt, Björn, Hartman, Johan, Haglund, Felix, Majellaro, Maria, Azuaje, Jhonny, Garcia-Mera, Xerardo, Brea, Jose M, Loza, Maria I, Jespers, Willem, Gutierrez-de-Teran, Hugo, Sotelo, Eddy, Lundqvist, Andreas
Опубликовано 2022Текст