Výsledky vyhledávání - Alejandra Tomás
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Disconnect between signalling potency and in vivo efficacy of pharmacokinetically optimised biased glucagon-like peptide-1 receptor agonists Autor Maria Lucey, Philip Pickford, Stavroula Bitsi, James Minnion, Jan Ungewiss, Katja Schoeneberg, Guy A. Rutter, Stephen R. Bloom, Alejandra Tomás, Ben Jones
Vydáno 2020Artigo -
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Abolishing β‐arrestin recruitment is necessary for the full metabolic benefits of G protein‐biased glucagon‐like peptide‐1 receptor agonists Autor Charlotte E. Hinds, Ellie Peace, Shiqian Chen, Iona Davies, Liliane El Eid, Alejandra Tomás, Tricia Tan, James Minnion, Ben Jones, Stephen R. Bloom
Vydáno 2023Artigo -
14
The Zinc Transporter Slc30a8/ZnT8 Is Required in a Subpopulation of Pancreatic α-Cells for Hypoglycemia-induced Glucagon Secretion Autor Antonia Solomou, Gargi Meur, Elisa A. Bellomo, David J. Hodson, Alejandra Tomás, Stéphanie Migrenne Li, Erwann Philippe, Pedro L. Herrera, Chr̀istophe Magnan, Guy A. Rutter
Vydáno 2015Artigo -
15
Divergent acute versus prolonged pharmacological GLP-1R responses in adult β cell–specific β-arrestin 2 knockout mice Autor Stavroula Bitsi, Liliane El Eid, Yusman Manchanda, Affiong I Oqua, Nimco Mohamed, Ben Hansen, Kinga Suba, Guy A. Rutter, Victoria Salem, Ben Jones, Alejandra Tomás
Vydáno 2023Artigo -
16
Binding Kinetics, Bias, Receptor Internalization and Effects on Insulin Secretion<i>in vitro</i>and<i>in vivo</i>of a Novel GLP-1R/GIPR Dual Agonist, HISHS-2001 Autor Yusman Manchanda, Ben Jones, Gaëlle Carrat, Zenouska Ramchunder, Piero Marchetti, Isabelle Leclerc, Rajamannar Thennati, Vinod Burade, Muthukumaran Natarajan, Pradeep Shahi, Alejandra Tomás, Guy A. Rutter
Vydáno 2025Pré-impressão -
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Biomimetic electromechanical stimulation to maintain adult myocardial slices in vitro Autor Samuel Watson, James Duff, Ifigeneia Bardi, Magdalena A. Zabielska-Kaczorowska, Santosh S. Atanur, Richard J. Jabbour, A. Simón, Alejandra Tomás, Ryszard T. Smoleński, Siân E. Harding, Filippo Perbellini, Cesare M. Terracciano
Vydáno 2019Artigo -
18
Signalling, trafficking and glucoregulatory properties of glucagon‐like peptide‐1 receptor agonists exendin‐4 and lixisenatide Autor Philip Pickford, Maria Lucey, Zijian Fang, Stavroula Bitsi, Jorge Bernardino de la Serna, Johannes Broichhagen, David J. Hodson, James Minnion, Guy A. Rutter, Stephen R. Bloom, Alejandra Tomás, Ben Jones
Vydáno 2020Artigo -
19
A Targeted RNAi Screen Identifies Endocytic Trafficking Factors That Control GLP-1 Receptor Signaling in Pancreatic β-Cells Autor Teresa Buenaventura, Nisha Kanda, Phoebe C. Douzenis, Ben Jones, Stephen R. Bloom, Pauline Chabosseau, Ivan R. Corrêa, Domenico Bosco, Lorenzo Piemonti, Piero Marchetti, Paul Johnson, A. M. James Shapiro, Guy A. Rutter, Alejandra Tomás
Vydáno 2017Artigo -
20
DRP1 levels determine the apoptotic threshold during embryonic differentiation through a mitophagy-dependent mechanism Autor Bárbara Pernaute, Salvador Pérez-Montero, Juan Miguel Sánchez Nieto, Aida Di Gregorio, Ana Lima, Katerina Lawlor, Sarah Bowling, Gianmaria Liccardi, Alejandra Tomás, Pascal Meier, Hiromi Sesaki, Guy A. Rutter, Ivana Barbaric, Tristan A. Rodríguez
Vydáno 2022Artigo
Vyhledávací nástroje:
Související témata
Biology
Cell biology
Endocrinology
Receptor
Biochemistry
Medicine
Chemistry
Internal medicine
Agonist
Diabetes mellitus
Type 2 diabetes
Insulin
Signal transduction
G protein-coupled receptor
Genetics
Glucagon-like peptide 1 receptor
Glucagon-like peptide-1
Endocytosis
Gene
Glucagon
Incretin
Internalization
Intracellular
Pharmacology
Secretion
Endocytic cycle
Endosome
Functional selectivity
In vivo
Arrestin